1. Signaling Pathways
  2. Neuronal Signaling
  3. Imidazoline Receptor
  4. Imidazoline Receptor Antagonist

Imidazoline Receptor Antagonist

Imidazoline Receptor Antagonists (3):

Cat. No. Product Name Effect Purity
  • HY-14561A
    Idazoxan hydrochloride
    Antagonist 99.32%
    Idazoxan hydrochloride (RX 781094 hydrochloride) is an α2-adrenoceptor antagonist and is also a imidazoline receptors (IRs) antagonist competitively antagonized the centrally induced hypotensive effect of imidazoline-like agents (IMs). Idazoxan hydrochloride also improves motor symptoms in Parkinson’s disease, L-DOPA-induced dyskinesias, and experimental Parkinsonism.
  • HY-101374A
    AGN 192403 hydrochloride
    Antagonist
    AGN 192403 (BRD4780) hydrochloride is an I1-Imidazoline receptor antagonist for cardiovascular and neurological research.
  • HY-B1416A
    Efaroxan hydrochloride
    Antagonist 99.94%
    Efaroxan hydrochloride is a potent, selective and orally active α2-adrenoceptor antagonist, with antidiabetic activity. Efaroxan hydrochloride is a selective I1-Imidazoline receptor antagonist. Efaroxan hydrochloride can be used for the research of cardiovascular disease.